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Results for "

congener

" in MedChemExpress (MCE) Product Catalog:

18

Inhibitors & Agonists

4

Natural
Products

Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-101139A
    Xanthine amine congener hydrochloride

    XAC hydrochloride

    		 Adenosine Receptor Neurological Disease
    Xanthine amine congener (XAC) hydrochloride is a non-selective adenosine receptor antagonist. Xanthine amine congener hydrochloride induces convulsions in mice .
    Xanthine amine <em>congener</em> hydrochloride
  • HY-128064
    Adenosine amine congener

    ADAC

    		 Adenosine Receptor Neurological Disease Inflammation/Immunology
    Adenosine amine congener (ADAC) is a selective A1 adenosine receptor agonist, can ameliorate noise- and Cisplatin-induced cochlear injury. Adenosine amine congener also has neuroprotective effects .
    Adenosine amine <em>congener</em>
  • HY-N0449
    Nordihydrocapsaicin

    		Others Others
    Nordihydrocapsaicin is a capsaicinoid analog and congener of capsaicin in chili peppers .
    Nordihydrocapsaicin
  • HY-101139
    Xanthine amine congener

    XAC

    		 Adenosine Receptor Neurological Disease
    Xanthine amine congener is a non-selective adenosine receptor antagonist . Xanthine amine congener induces convulsions in mice .
    Xanthine amine <em>congener</em>
  • HY-110303
    Xanthine amine congener dihydrochloride

    XAC dihydrochloride

    		 Adenosine Receptor Neurological Disease
    Xanthine amine congener dihydrochloride (XAC dihydrochloride) is a potent Adenosine A1 receptor and A2 receptor antagonist with IC50 values of 1.8 and 114 nM, respectively. Xanthine amine congener acts as a convulsant agent in mice model .
    Xanthine amine <em>congener</em> dihydrochloride
  • HY-N12760
    Lobophorin CR-2

    		Others Cancer
    Lobophorin CR-2 is a lobophorin congener which induces UPR-associated gene expression, inhibits oral squamous cell carcinoma cell growth, and causes UPR-dependent cell death in MEF cells .
    Lobophorin CR-2
  • HY-117765
    RS-5773

    		Calcium Channel Neurological Disease
    RS-5773 is a calcium channel inhibitor and a diltiazem congener. RS-5773 has antianginal effect and does not cause excessive hypotension or depression of atrioventricular conduction .
    RS-5773
  • HY-148649
    Demethyl bleomycin A2

    		Antibiotic Others
    Demethyl bleomycin A2 is a Bleomycin (HY-108345) congener. The DNA cleavage of demethyl bleomycin A2 is insensitive to the presence of 5-Methylcytidine (HY-113135) .
    Demethyl bleomycin A2
  • HY-W013788
    2-Palmitoylglycerol

    2-Palm-Gl

    		 Cannabinoid Receptor Neurological Disease
    2-Palmitoylglycerol (2-Palm-Gl), an congener of 2-arachidonoylglycerol (2-AG), is a modest cannabinoid receptor CB1 agonist. 2-Palmitoylglycerol also may be an endogenous ligand for GPR119 .
    2-Palmitoylglycerol
  • HY-144893
    OKI-006

    		HDAC Cancer
    OKI-006 is a potent and orally active inhibitor of histone deacetylase (HDAC). OKI-006 is a unique congener of the natural product HDAC inhibitor largazole. Histone deacetylases (HDACs) play critical roles in epigenomic regulation, and histone acetylation is dysregulated in many human cancers. OKI-006 has the potential for the research of cancer disease .
    OKI-006
  • HY-105890
    Spiroplatin

    TNO 6

    		 Others Cancer
    Spiroplatin is a Cisplatin (HY-17394) congener and has antitumor activity .
    Spiroplatin
  • HY-146970
    Lankacyclinone C

    		Antibiotic Cancer
    Lankacyclinone C is a lankacidin C congener lacking the δ-lactone moiety, with antitumor activity .
    Lankacyclinone C
  • HY-N0685
    Pseudohypericin

    		HIV Infection
    Pseudohypericin and its congener Hypericin are the major hydroxylated phenanthroperylenediones present in Hypericum species. Pseudohypericin shows anti-HIV activity .
    Pseudohypericin
  • HY-W140555
    5,7-Dimethoxyphthalide

    		Others Others
    5,7-Dimethoxyphthalide can be conjugated to functionalized long-chain alkyl iodides that are useful in designing a focused mini-library of analogous and congeners of CJ-molecules for SAR study .
    5,7-Dimethoxyphthalide
  • HY-146102
    M1 ligand 1

    		mAChR Others
    M1 ligand 1 (compound 3b-b) is a muscarinic acetylcholine receptor M1 ligand. M1 ligand 1 is a N-desmethyl congener of arecoline derivative. M1 ligand 1 can be used as PET (positron emission tomography) radiotracer .
    M1 ligand 1
  • HY-129454
    TPU-0037A

    Antibiotic TPU-0037-A

    		 Others Infection
    TPU-0037A is an antibiotic and a congener of lydicamycin. It inhibits the growth of Gram-positive bacteria, including methicillin-resistant S. aureus (MRSA), B. subtilis, and M. luteus (MICs=1.56-12.5 μg/mL), but not Gram-negative E. coli, P. mirabilis, P. vulgaris, or P. aeruginosa strains (MICs=>50 μg/mL).
    TPU-0037A
  • HY-144286
    CXCR4 antagonist 3

    		CXCR Infection
    CXCR4 antagonist 3 (compound 12a) is a potent antagonist of CXCR4 with an IC50 of 11 nM. CXCR4 antagonist 3 is a congener of TIQ15. CXCR4 antagonist 3 demonstrates the best overall properties including CXCR4 antagonism, CYP 2D6 inhibition, metabolic stability, and permeability. CXCR4 antagonist 3 has the potential for the research of human immunodeficiency virus .
    CXCR4 antagonist 3
  • HY-118816
    11β-Prostaglandin F2α

    11-epi PGF2α-EA; 11β-PGF2α-EA; 11β-Prostamide F2α

    		 Others Metabolic Disease
    11β-Prostaglandin F2α ethanolamide (11β-PGF2α-EA) is the theoretical hepatic metabolite of PGD2-EA, produced during COX-2 metabolism of the endogenous cannabinoid AEA which is found in brain, liver, and other mammalian tissues.1 AEA can be used directly by COX-2 and specific PG synthase to produce ethanolamide congeners of the classical PGs. PGD2-EA is formed in activated RAW 264.7 cells treated with AEA.
    11β-Prostaglandin F2α

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